SCHEMBL5251237

SCHEMBL5251237

CCN1CCN(c2ccc(-c3cn4cccc(OC(N)=O)c4n3)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 6/20 0.44
SYK P43405 1/20 0.42
DRD2 P14416 2/20 0.42
DRD3 P35462 2/20 0.42
DHODH Q02127 1/20 0.40
HRH3 Q9Y5N1 2/20 0.40
ALDH1A1 P00352 2/20 0.39
ALDH1A2 O94788 1/20 0.39
ALDH1A3 P47895 1/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
HTR2A P28223 1/20 0.39
LMNA P02545 1/20 0.39
MEN1 O00255 1/20 0.39
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5250582 0.92 DRD2 (0.45) GNRHRDRD2DRD3DHODHHRH3
SCHEMBL5251170 0.91 DRD2 (0.47) GNRHRDRD2DRD3HRH3KDM4E
SCHEMBL5256363 0.89 CHEK1 (0.47) DRD2DRD3DHODHHRH3ALDH1A1
SCHEMBL5329494 0.88 DRD4 (0.43) GNRHRDRD2DRD3DHODHALDH1A1
SCHEMBL5253308 0.88 HRH3 (0.45) GNRHRDRD2DRD3HRH3HTR2A
SCHEMBL5255275 0.86 TLR9 (0.46) DHODHHRH3ALDH1A1ALDH1A2ALDH1A3
SCHEMBL5248611 0.85 CHEK1 (0.44) SYKDRD2DRD3DHODHHRH3
SCHEMBL5248183 0.85 TLR9 (0.42) DHODHALDH1A1ALDH1A2ALDH1A3KDM4E
SCHEMBL5076308 0.85 DHODH (0.50) GNRHRSYKDHODHHRH3ALDH1A1
SCHEMBL5300289 0.85 DGAT1 (0.42) GNRHRDRD2DRD3DHODHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1257551-B1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2007-09-05 EP disclosed