SCHEMBL5329494

SCHEMBL5329494

NC(=O)Oc1cccn2cc(-c3ccc(N4CCN(Cc5ccccc5)CC4)cc3)nc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
HTR2A P28223 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
DHODH Q02127 1/20 0.43
GNRHR P30968 3/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5300289 0.96 DGAT1 (0.42) DRD4MAPTTSHRMAPK1HTR2A
SCHEMBL5251237 0.88 GNRHR (0.44) MAPTHTR2ADHODHGNRHRKDM4E
SCHEMBL5250582 0.86 DRD2 (0.45) HTR2ADHODHGNRHRDRD2DRD3
SCHEMBL5076369 0.86 DHODH (0.53) DRD4MAPTTSHRMAPK1HTR2A
SCHEMBL5256363 0.84 CHEK1 (0.47) MAPTDHODHKDM4EALDH1A1DRD2
SCHEMBL5251170 0.84 DRD2 (0.47) HTR2AGNRHRKDM4EDRD2DRD3
SCHEMBL5077273 0.83 DHODH (0.49) DRD4HTR2AHDAC3HDAC4HDAC1
SCHEMBL5248183 0.82 TLR9 (0.42) TSHRDHODHKDM4EALDH1A1
SCHEMBL5255275 0.82 TLR9 (0.46) MAPTDHODHKDM4EALDH1A1
SCHEMBL5253308 0.81 HRH3 (0.45) HTR2AGNRHRDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1257551-B1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2007-09-05 EP disclosed