SCHEMBL5251986

SCHEMBL5251986

Cc1c(CC(=O)O)c2cnccc2n1Cc1ccc(F)c(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 13/20 0.53
LMNA P02545 2/20 0.53
CYP1A2 P05177 2/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2C9 P11712 2/20 0.53
TSHR P16473 2/20 0.53
CYP2C19 P33261 2/20 0.53
PMP22 Q01453 2/20 0.53
MEN1 O00255 1/20 0.53
RGS12 O14924 1/20 0.53
ALDH1A1 P00352 1/20 0.53
MAPT P10636 1/20 0.53
PKM P14618 1/20 0.53
NFKB1 P19838 1/20 0.53
MAPK1 P28482 1/20 0.53
GNAI1 P63096 1/20 0.53
KMT2A Q03164 1/20 0.53
HIF1A Q16665 1/20 0.53
KDM4E B2RXH2 1/20 0.52
BLM P54132 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5250503 0.82 PTGDR2 (0.64) PTGDR2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL5248719 0.81 PTGDR2 (0.54) PTGDR2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL1939490 0.80 PTGDR2 (0.83) PTGDR2
SCHEMBL2005651 0.78 LMNA (0.64) PTGDR2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL2996259 0.75 PTGDR2 (0.60) PTGDR2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL5454133 0.73 LMNA (0.63) PTGDR2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL13802405 0.73 PTGDR2 (0.70) PTGDR2PTGESALOX5PLA2G1BPLA2G2A
SCHEMBL2005008 0.73 LMNA (0.59) PTGDR2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL3003631 0.72 LMNA (0.68) PTGDR2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL4209387 0.72 PTGDR2 (0.74) PTGDR2LMNACYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761529-A2 PYRROLOPYRIDINE DERIVATIVES AND THEIR USE AS CRTH2 ANTAGONISTS Novartis AG (CH) 2007-03-14 EP claimed
WO-2005123731-A2 PYRROLOPYRIDINE DERIVATIVES AND THEIR USE AS CRTH2 ANTAGONISTS NOVARTIS AG (CH) 2005-12-29 WO claimed