SCHEMBL525259

SCHEMBL525259

NCC(c1ccccc1)N(CCO)CCO

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.45
HTR2A P28223 3/20 0.45
SLC6A4 P31645 4/20 0.41
SLC6A2 P23975 3/20 0.41
SLC6A3 Q01959 2/20 0.40
GABBR2 O75899 2/20 0.39
GABBR1 Q9UBS5 2/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
HRH1 P35367 2/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
GAA P10253 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11401685 0.79 KMT2A (0.36) HTR2AHRH1MEN1KMT2AGAA
SCHEMBL15152279 0.77 CYP2C19 (0.46) HTR2AHRH1MEN1KMT2AGAA
SCHEMBL17803383 0.76 TAAR1 (0.48) TAAR1HTR2ASLC6A4SLC6A2SLC6A3
SCHEMBL24885673 0.75 OPRD1 (0.41) HTR2AHRH1MEN1KMT2AALDH1A1
SCHEMBL11173715 0.75 MEN1 (0.40) TAAR1HTR2AHRH1MEN1KMT2A
SCHEMBL11094516 0.74 TAAR1 (0.46) TAAR1HTR2ASLC6A4SLC6A2SLC6A3
SCHEMBL11701106 0.74 NR1H2 (0.43) HTR2AHRH1MEN1KMT2AALDH1A1
SCHEMBL3931089 0.72 TRPA1 (0.48) HTR2AHRH1MEN1KMT2AALDH1A1
Trolamine SCHEMBL21177786 0.72 TAAR1 (0.47) TAAR1HTR2ASLC6A4SLC6A2SLC6A3
SCHEMBL7093914 0.71 TAAR1 (0.52) TAAR1HTR2ASLC6A4SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2598142-A1 DIPHENYL ETHER COMPOUNDS FOR THE TREATMENT OF LIVER, LUNG DISORDERS, DIABETIC COMPLICATIONS AND CARDIOVASCULAR DISEASES Orchid Chemicals and Pharmaceuticals Ltd (IN) 2013-06-05 EP disclosed
WO-2012014218-A1 DIPHENYL ETHER COMPOUNDS FOR THE TREATMENT OF LIVER, LUNG DISORDERS, DIABETIC COMPLICATIONS AND CARDIOVASCULAR DISEASES ORCHID RESEARCH LABORATORIES LTD. (IN) 2012-02-02 WO disclosed