SCHEMBL5254657

SCHEMBL5254657

CCc1cc(Nc2cc(C)n[nH]2)nc(-c2ccccc2OF)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.35
KDM4E B2RXH2 6/20 0.35
MAPK1 P28482 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ADORA3 P0DMS8 3/20 0.34
ADORA1 P30542 2/20 0.34
MEN1 O00255 7/20 0.34
KMT2A Q03164 7/20 0.34
HSD17B10 Q99714 5/20 0.34
ALOX15 P16050 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HPGD P15428 2/20 0.34
HTT P42858 3/20 0.33
NPSR1 Q6W5P4 3/20 0.33
ATM Q13315 2/20 0.33
PDE4B Q07343 2/20 0.33
RECQL P46063 1/20 0.33
BRD4 O60885 1/20 0.33
TSHR P16473 3/20 0.32
CYP1A2 P05177 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL786116 0.89 TRPA1 (0.36) MAPTKDM4EMAPK1L3MBTL1NPSR1
SCHEMBL786645 0.82 ABCG2 (0.47) MAPTL3MBTL1MEN1KMT2ANPSR1
SCHEMBL786451 0.77 NPC1 (0.41) ADORA3ADORA1MEN1KMT2APDE4B
SCHEMBL5256614 0.76 ABCG2 (0.44) MAPTKDM4EMAPK1L3MBTL1MEN1
SCHEMBL786316 0.76 PDE4B (0.43) ADORA3SMN1; SMN2PDE4BCYP1A2CYP3A4
SCHEMBL786879 0.75 ADORA3 (0.40) MAPTADORA3PDE4BCYP1A2
SCHEMBL2205769 0.72 RAB9A (0.43) MAPTKDM4EL3MBTL1MEN1KMT2A
SCHEMBL786491 0.72 MEN1 (0.58) MAPTL3MBTL1MEN1KMT2ASMN1; SMN2
SCHEMBL2203919 0.71 COMT (0.35) MAPTKDM4EMEN1KMT2AHSD17B10
SCHEMBL2204725 0.71 FFAR1 (0.36) MAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318814-B1 TRIAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2007-05-30 EP disclosed