SCHEMBL5255103

SCHEMBL5255103

COC(=O)[C@H](Cc1ccc(Oc2nccc3cnccc23)cc1)NS(=O)(=O)N1C(C)CCCC1C

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.37
F2 P00734 8/20 0.35
PRSS1 P07477 3/20 0.35
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
SCN5A Q14524 1/20 0.33
SCN9A Q15858 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33
ITGB7 P26010 1/20 0.33
TRPV1 Q8NER1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225880 0.94 P2RX7 (0.38) P2RX7F2PRSS1ALDH1A1TP53
SCHEMBL5258334 0.86 NAMPT (0.36) P2RX7F2PRSS1ALDH1A1TP53
SCHEMBL5256634 0.83 CYP1A2 (0.38) P2RX7F2PRSS1SMN1; SMN2CYP3A4
SCHEMBL5259948 0.81 P2RX7 (0.38) P2RX7ALDH1A1SMN1; SMN2CYP3A4CYP2C9
SCHEMBL5256327 0.81 P2RX7 (0.37) P2RX7CYP3A4CYP2C9SCN5ASCN9A
SCHEMBL5255111 0.79 P2RX7 (0.34) P2RX7ALDH1A1TP53SMN1; SMN2CYP3A4
SCHEMBL5257627 0.79 CA12 (0.37) P2RX7CYP3A4CYP2C9SCN5ASCN9A
SCHEMBL5227174 0.78 NAMPT (0.37) P2RX7F2ALDH1A1TP53SMN1; SMN2
SCHEMBL5224364 0.76 CYP1A2 (0.39) P2RX7F2PRSS1SMN1; SMN2CYP3A4
SCHEMBL5227139 0.75 ITGB1 (0.41) P2RX7ALDH1A1SMN1; SMN2ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622867-B1 N-(2-PHENYLETHYL)SULFAMIDE DERIVATIVES AS INTEGRIN ALPHA4 ANTAGONISTS ALMIRALL LAB (ES) 2007-09-19 EP claimed