SCHEMBL5255111

SCHEMBL5255111

CC1CCCC(C)N1S(=O)(=O)N[C@@](C)(Cc1ccc(Oc2nccc3cnccc23)cc1)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 9/20 0.34
FFAR1 O14842 1/20 0.33
NAMPT P43490 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TRPV1 Q8NER1 4/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5258338 0.85 NAMPT (0.37) NAMPTALDH1A1TP53SMN1; SMN2TRPV1
SCHEMBL5225880 0.82 P2RX7 (0.38) P2RX7ALDH1A1TP53SMN1; SMN2
SCHEMBL5256637 0.82 CYP3A4 (0.37) P2RX7FFAR1SMN1; SMN2TRPV1CYP3A4
SCHEMBL5259953 0.81 FFAR1 (0.36) P2RX7FFAR1ALDH1A1SMN1; SMN2TRPV1
SCHEMBL5256333 0.80 FFAR1 (0.37) P2RX7FFAR1ALDH1A1SMN1; SMN2TRPV1
SCHEMBL5255103 0.79 P2RX7 (0.37) P2RX7ALDH1A1TP53SMN1; SMN2TRPV1
SCHEMBL5257628 0.78 CYP3A4 (0.36) P2RX7FFAR1ALDH1A1SMN1; SMN2TRPV1
SCHEMBL5182529 0.76 LATS1 (0.40) P2RX7FFAR1TRPV1
SCHEMBL5307756 0.70 ITGA4 (0.44)
SCHEMBL7107376 0.70 ITGB1 (0.36) FFAR1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622867-B1 N-(2-PHENYLETHYL)SULFAMIDE DERIVATIVES AS INTEGRIN ALPHA4 ANTAGONISTS ALMIRALL LAB (ES) 2007-09-19 EP claimed