SCHEMBL5255182

SCHEMBL5255182

NC(=O)Oc1cccn2cc(-c3ccc(N4CCCNCC4)cc3)nc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 5/20 0.40
TLR9 Q9NR96 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
SCN9A Q15858 1/20 0.39
DHODH Q02127 1/20 0.39
MAPKAPK2 P49137 1/20 0.38
CREBBP Q92793 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
PIM1 P11309 3/20 0.37
PIM3 Q86V86 3/20 0.37
PIM2 Q9P1W9 2/20 0.37
ACVR1 Q04771 2/20 0.37
SUV39H2 Q9H5I1 1/20 0.37
TGFBR1 P36897 1/20 0.36
ALDH1A2 O94788 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ALDH1A3 P47895 1/20 0.36
CDK4 P11802 1/20 0.36
CCND3 P30281 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5248183 0.96 TLR9 (0.42) TLR9TLR7SCN9ADHODHMAPKAPK2
SCHEMBL5073422 0.85 DHODH (0.49) ATRDHODHMAPKAPK2CREBBPCHRNB2
SCHEMBL5248611 0.85 CHEK1 (0.44) DHODHCREBBPPIM1PIM3PIM2
SCHEMBL5256363 0.84 CHEK1 (0.47) DHODHPIM1PIM3PIM2ACVR1
SCHEMBL5255275 0.82 TLR9 (0.46) TLR9TLR7DHODHACVR1TGFBR1
SCHEMBL5251237 0.82 GNRHR (0.44) DHODHALDH1A2ALDH1A1ALDH1A3
SCHEMBL5073335 0.81 DHODH (0.53) TLR9TLR7SCN9ADHODHMAPKAPK2
SCHEMBL5300289 0.80 DGAT1 (0.42) DHODHALDH1A1PARP1
SCHEMBL5250582 0.80 DRD2 (0.45) DHODH
SCHEMBL5253308 0.79 HRH3 (0.45) CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1257551-B1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2007-09-05 EP disclosed