SCHEMBL525885

SCHEMBL525885

C=CCc1ccc(OC)c(-c2cc(CC=C)ccc2OC(CCCl)c2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 6/20 0.52
GABRB2 P47870 6/20 0.52
ALOX5 P09917 6/20 0.47
CNR2 P34972 2/20 0.47
ALDH1A1 P00352 4/20 0.47
PPARG P37231 1/20 0.47
PPARD Q03181 1/20 0.47
PPARA Q07869 1/20 0.47
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
CYP3A4 P08684 3/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
HTT P42858 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL525549 0.87 SLC6A4 (0.59) GABRA1GABRB2ALOX5CNR2ALDH1A1
Hydrochloric Acid SCHEMBL725835 0.86 SLC6A2 (0.60) GABRA1GABRB2ALOX5CNR2ALDH1A1
SCHEMBL14125144 0.77 GABRA1 (0.81) GABRA1GABRB2ALOX5CNR2ALDH1A1
SCHEMBL9404982 0.76 ALDH1A1 (0.58) GABRA1GABRB2ALOX5ALDH1A1PPARG
SCHEMBL525899 0.76 SLC6A4 (0.52) GABRA1GABRB2MEN1KMT2ACYP3A4
SCHEMBL525534 0.76 GABRA1 (0.54) GABRA1GABRB2ALOX5CNR2ALDH1A1
Hydrochloric Acid SCHEMBL530274 0.75 GABRA1 (0.53) GABRA1GABRB2ALOX5CNR2ALDH1A1
Hydrochloric Acid SCHEMBL726060 0.75 SLC6A4 (0.51) GABRA1GABRB2MEN1KMT2ACYP3A4
SCHEMBL526216 0.75 SLC6A4 (0.48) ALDH1A1MEN1KMT2ACYP3A4HTT
SCHEMBL9772801 0.74 SLC6A2 (0.68) MEN1KMT2ACYP3A4LMNASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP disclosed
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP disclosed
WO-2012013691-A1 MULTITARGET SUBSTITUTED BIPHENYL DIOL DERIVATIVES PROUS INSTITUTE FOR BIOMEDICAL RESEARCH, S.A. (ES) 2012-02-02 WO disclosed
WO-2012013691-A1 MULTITARGET SUBSTITUTED BIPHENYL DIOL DERIVATIVES PROUS INSTITUTE FOR BIOMEDICAL RESEARCH, S.A. (ES) 2012-02-02 WO disclosed