SCHEMBL5259159

SCHEMBL5259159

O=C(O)Nc1nccc2[nH]ccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.39
PIK3C3 Q8NEB9 2/20 0.39
TRPA1 O75762 2/20 0.38
GSK3B P49841 3/20 0.37
GSK3A P49840 1/20 0.37
JAK2 O60674 2/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
IKBKB O14920 2/20 0.36
CHUK O15111 2/20 0.36
DRD1 P21728 1/20 0.36
PRKCI P41743 2/20 0.36
AXL P30530 1/20 0.36
AURKB Q96GD4 2/20 0.36
DAPK3 O43293 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
CSF1R P07333 1/20 0.36
RET P07949 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14062242 0.85 PIK3C3 (0.49) NUDT1PIK3C3TRPA1JAK3DYRK1A
SCHEMBL14059926 0.83 NUDT1 (0.40) NUDT1PIK3C3TRPA1GSK3BGSK3A
SCHEMBL15753484 0.81 HPGDS (0.47) NUDT1PIK3C3GSK3BGSK3AJAK2
SCHEMBL3887252 0.81 NUDT1 (0.51) NUDT1KDRMAPK1
SCHEMBL15753311 0.80 GSK3B (0.55) GSK3BGSK3AJAK2TYK2PRKCI
SCHEMBL13759613 0.78 ATR (0.42) NUDT1PIK3C3JAK2JAK1TYK2
SCHEMBL23877021 0.75 TRPA1 (0.45) TRPA1JAK2IKBKBCHUKDRD1
Hydrochloric Acid SCHEMBL29243587 0.74 TRPA1 (0.44) TRPA1JAK2IKBKBCHUKDRD1
SCHEMBL9936674 0.74 PDE3B (0.42) NUDT1PIK3C3TRPA1JAK2IKBKB
SCHEMBL21603403 0.72 DRD1 (0.39) NUDT1TRPA1DRD1PRKCIAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742948-A2 BICYCLIC HETEROCYCLES AS KINASE INHIBITORS Bristol-Myers Squibb Company (US) 2007-01-17 EP disclosed
WO-2005116028-A2 BICYCLIC HETEROCYCLES AS KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-12-08 WO disclosed