SCHEMBL5259605

SCHEMBL5259605

Fc1ccccc1-c1nc(Nc2n[nH]c3ccccc23)cc(C2CCCCC2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.48
GSK3B P49841 2/20 0.48
GBA1 P04062 1/20 0.43
FADS1 O60427 2/20 0.41
LCK P06239 1/20 0.40
ITK Q08881 1/20 0.40
AURKB Q96GD4 1/20 0.40
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
ADRA2A P08913 2/20 0.36
TRPA1 O75762 1/20 0.36
GRM4 Q14833 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA2A P29274 2/20 0.35
EGFR P00533 1/20 0.35
USP1 O94782 1/20 0.35
WDR48 Q8TAF3 1/20 0.35
PLK4 O00444 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL786010 0.87 USP1 (0.49) GSK3AGSK3BFADS1LCKITK
SCHEMBL13854193 0.82 LCK (0.39) GSK3AGSK3BFADS1LCKITK
SCHEMBL958497 0.82 CYP1A2 (0.43) GSK3AGSK3BFADS1LCKITK
SCHEMBL12653894 0.79 MAPK8 (0.38) GSK3AGSK3BFADS1LCKITK
SCHEMBL801495 0.79 CYP1A2 (0.48) LCKITKAURKBUSP1WDR48
SCHEMBL5261414 0.78 WNT1 (0.45) FADS1POLBMAPTMAPK1ADRA2A
SCHEMBL801908 0.76 USP1 (0.41) GSK3AGSK3BFADS1LCKITK
SCHEMBL786816 0.76 USP1 (0.43) FADS1LCKITKAURKBMAPT
SCHEMBL801899 0.75 USP1 (0.40) GSK3AGSK3BFADS1LCKITK
SCHEMBL801905 0.74 RBP4 (0.46) LCKITKAURKBGRM4EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318814-B1 TRIAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2007-05-30 EP disclosed