SCHEMBL5260599

SCHEMBL5260599

c1ccc2c(c1)OC1COCCC21

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
CHRNB4 P30926 2/20 0.36
CHRNA3 P32297 2/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
LMNA P02545 2/20 0.32
CRHBP P24387 2/20 0.32
CRHR2 Q13324 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
HTT P42858 1/20 0.32
CYP3A4 P08684 1/20 0.32
IDO1 P14902 1/20 0.32
TDO2 P48775 1/20 0.32
HTR6 P50406 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26227708 0.79 ESR1 (0.42) ESR1ESR2CHRNB4CHRNA3CHRNB2
SCHEMBL8515749 0.77 CYP19A1 (0.40)
SCHEMBL7317272 0.76 ESR1 (0.47) ESR1ESR2CHRNB4CHRNA3CHRNB2
SCHEMBL10682685 0.76 ESR1 (0.51) ESR1ESR2CHRNB4CHRNA3CHRNB2
SCHEMBL9391610 0.76 ESR1 (0.47) ESR1ESR2CHRNB4CHRNA3CHRNB2
SCHEMBL17974163 0.72 ESR1 (0.40) ESR1ESR2DRD2DRD3HTR6
SCHEMBL20045526 0.70 HTR6 (0.58) HTR6
SCHEMBL2226246 0.70 HTR6 (0.58) HTR6
Hydrochloric Acid SCHEMBL2223844 0.69 HTR6 (0.60) HTR6
SCHEMBL9910980 0.68 SIGMAR1 (0.48) CHRNB4CHRNA3CHRNB2CHRNA4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778680-A2 SPIROCYCLIC CYCLOHEXANE DERIVATIVES Grünenthal GmbH (DE) 2007-05-02 EP disclosed
WO-2006018184-A2 SPIROCYCLIC CYCLOHEXANE DERIVATIVES Grünenthal GmbH (DE) 2006-02-23 WO disclosed