SCHEMBL8515749

SCHEMBL8515749

O=C1c2ccccc2OC2COCCC12

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.40
MAOB P27338 3/20 0.37
ADORA3 P0DMS8 2/20 0.37
AR P10275 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HSD17B10 Q99714 1/20 0.37
RET P07949 1/20 0.36
KDR P35968 1/20 0.36
SIGMAR1 Q99720 2/20 0.36
STK17B O94768 1/20 0.35
HSD11B1 P28845 1/20 0.33
AKR1C3 P42330 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878141 0.88 CYP19A1 (0.40) CYP19A1MAOBADORA3ARKDM4E
SCHEMBL8534500 0.80 PBRM1 (0.43) CYP19A1AR
SCHEMBL9882174 0.80 PBRM1 (0.43) CYP19A1AR
SCHEMBL8534502 0.80 PBRM1 (0.43) CYP19A1AR
SCHEMBL5260599 0.77 ESR1 (0.38)
SCHEMBL877529 0.73 ADORA3 (0.33) CYP19A1MAOBADORA3ARKDM4E
SCHEMBL25079067 0.72 CYP19A1 (0.50) CYP19A1MAOBSIGMAR1
SCHEMBL15287877 0.70 ADORA3 (0.36) CYP19A1MAOBADORA3ARKDM4E
SCHEMBL28984669 0.70 MAOB (0.49) CYP19A1MAOBADORA3ARKDM4E
SCHEMBL11381317 0.69 SIGMAR1 (0.60) CYP19A1MAOBADORA3ARKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071458-A1 HETEROCYCLIC INHIBITORS OF BETA - SECRETASE FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES ARRAY BIOPHARMA INC. (US) 2012-05-31 WO disclosed