SCHEMBL5261114

SCHEMBL5261114

COc1cc(C(C(=O)O)N(CC(=O)OC(C)(C)C)C(=O)C(F)(F)F)cc(OC)n1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 15/20 0.33
EDNRA P25101 15/20 0.33
CASR P41180 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
STING1 Q86WV6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5186385 0.89 EDNRB (0.32) EDNRBEDNRA
SCHEMBL5259046 0.87 EDNRB (0.36) EDNRBEDNRAKDM4EALDH1A1
SCHEMBL5313941 0.85 EDNRB (0.34) EDNRBEDNRAKDM4EALDH1A1
SCHEMBL4694873 0.75 NR1D1 (0.34) MTNR1AMTNR1B
SCHEMBL4693024 0.72
SCHEMBL5255513 0.69 CASR (0.43) CASRALDH1A1
SCHEMBL5252254 0.69 KDM4E (0.39) EDNRBEDNRAKDM4EALDH1A1MTNR1A
SCHEMBL24326337 0.68 REN (0.37) CASRALDH1A1
SCHEMBL4145065 0.67 NR1D1 (0.33) ALDH1A1MTNR1AMTNR1B
SCHEMBL899172 0.64 KDM4E (0.40) EDNRBEDNRACASRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed