SCHEMBL5259046

SCHEMBL5259046

COc1cc(C(C(=O)O)N(CC(=O)O)C(=O)C(F)(F)F)cc(OC)n1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 16/20 0.36
EDNRA P25101 16/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
LMNA P02545 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5313941 0.90 EDNRB (0.34) EDNRBEDNRAKDM4EALDH1A1NR1H2
SCHEMBL5261114 0.87 EDNRB (0.33) EDNRBEDNRAKDM4EALDH1A1
SCHEMBL5186385 0.76 EDNRB (0.32) EDNRBEDNRA
SCHEMBL25254031 0.65 ALOX5 (0.42) NR1H2NR1H3
SCHEMBL25296546 0.65 ALOX5 (0.42) NR1H2NR1H3
SCHEMBL4692611 0.65 NR1H2 (0.30) NR1H2NR1H3
SCHEMBL29002093 0.64 AKR1C3 (0.54) EDNRBEDNRAKDM4EALDH1A1LMNA
SCHEMBL5258507 0.64 TSHR (0.50) EDNRBEDNRAKDM4EALDH1A1LMNA
SCHEMBL5252111 0.63 KMT2A (0.43) ALDH1A1NR1H2NR1H3
SCHEMBL8986465 0.62 PKM (0.41) KDM4EALDH1A1LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed