SCHEMBL5261284

SCHEMBL5261284

COc1ccc2[nH]c(S(=O)(=O)c3ccccc3)c(Br)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
MAPT P10636 5/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
KDM4E B2RXH2 3/20 0.49
HPGD P15428 3/20 0.49
HSD17B10 Q99714 2/20 0.49
ABCG2 Q9UNQ0 1/20 0.48
GFER P55789 2/20 0.47
TSHR P16473 1/20 0.47
GAA P10253 3/20 0.44
ADORA2B P29275 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
POLB P06746 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19717983 0.83 ALDH1A1 (0.52) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL19717747 0.80 GAA (0.45) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL5263730 0.80 MEN1 (0.44) ALDH1A1MEN1KMT2AKDM4EHSD17B10
SCHEMBL11015974 0.80 CA2 (0.47) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL3647177 0.78 HTR6 (0.43) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL19718029 0.77 ALDH1A1 (0.43) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL9737712 0.76 ALDH1A1 (0.49) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL19717746 0.76 SMN1; SMN2 (0.52) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL5784803 0.73 MAPT (0.78) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL19717957 0.72 ALDH1A1 (0.54) ALDH1A1MAPTMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3468950-A1 AZA-TANSHINONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THERAPY Universita' degli Studi di Milano (IT) 2019-04-17 EP disclosed
WO-2017216732-A1 AZA-TANSHINONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THERAPY UNIVERSITA' DEGLI STUDI DI MILANO (IT) 2017-12-21 WO disclosed
EP-1786813-A2 BICYCLIC HETEROARYL PDE4B INHIBITORS PLEXXIKON, INC. (US) 2007-05-23 EP disclosed
WO-2006026754-A9 BICYCLIC HETEROARYL PDE4B INHIBITORS PLEXXIKON INC (US) 2006-04-20 WO disclosed
WO-2006026754-A2 BICYCLIC HETEROARYL PDE4B INHIBITORS PLEXXIKON, INC. (US) 2006-03-09 WO disclosed