SCHEMBL5262287

SCHEMBL5262287

Nc1cc(O)nc(-c2ccccc2)n1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.66
ADORA1 P30542 7/20 0.66
ADORA3 P0DMS8 3/20 0.52
ADORA2B P29275 3/20 0.52
POLB P06746 1/20 0.52
KMT2A Q03164 7/20 0.48
MEN1 O00255 6/20 0.48
ALDH1A1 P00352 4/20 0.48
MAPT P10636 3/20 0.48
HPGD P15428 3/20 0.48
NTSR1 P30989 1/20 0.48
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
HTT P42858 1/20 0.47
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.42
GLA P06280 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NOTUM Q6P988 1/20 0.41
HSP90AA1 P07900 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720836 0.85 ADORA2A (0.79) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL18760499 0.85 MEN1 (0.57) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL3165362 0.85 MEN1 (0.57) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL6038198 0.84 ADORA2A (0.46) ADORA2AADORA1ADORA2BKMT2AMEN1
SCHEMBL2118725 0.81 MEN1 (0.59) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL1490059 0.79 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL3307656 0.79 MEN1 (0.68) ADORA2AADORA1ADORA3ADORA2BKMT2A
SCHEMBL13933596 0.76 ADORA2A (0.66) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL19417188 0.76 ADORA2A (0.92) ADORA2AADORA1ADORA3ADORA2BPOLB
SCHEMBL3156245 0.76 ADORA2A (0.66) ADORA2AADORA1ADORA3ADORA2BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794135-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE Amgen Inc. (US) 2007-06-13 EP disclosed
WO-2006037117-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE AMGEN INC. (US) 2006-04-06 WO disclosed
US-20060069110-A1 Substituted heterocyclic compounds and methods of use AMGEN INC. 2006-03-30 US disclosed
EP-0297397-B1 PREPARATION OF DIAZO AND AZO COMPOUNDS BAYER AG (DE) 1993-08-04 EP disclosed
US-4942225-A Preparation of diazo and azo compounds using azidoformamidium salts BAYER AKTIENGESELLSCHAFT (DE) 1990-07-17 US disclosed
EP-0218206-B1 DISAZO PIGMENTS HAVING A PIPERAZINE BRIDGING MEMBER BASF Aktiengesellschaft (DE) 1990-02-07 EP disclosed
EP-0297397-A2 Preparation of diazo and azo compounds BAYER AG (DE) 1989-01-04 EP disclosed
US-4764599-A INK PIGMENTS, SURFACE COATING, PLASTICS-SULFUR-FREE BASF AKTIENGESELLSCHAFT (DE) 1988-08-16 US disclosed
EP-0120255-B1 REACTIVE DYES BAYER AG (DE) 1987-04-15 EP disclosed
EP-0218206-A2 Disazo pigments having a piperazine bridging member BASF Aktiengesellschaft (DE) 1987-04-15 EP disclosed
US-4556707-A DYEING CELLULOSE FIBERS AND POLYAMIDE FIBERS BAYER AKTIENGESELLSCHAFT (DE) 1985-12-03 US disclosed
EP-0073463-B1 INSERTION COMPOUNDS, INTERCALATION COMPOUNDS AND SOLID SOLUTIONS OF COLOURED METALLIC ORGANIC DERIVATIVES BAYER AG (DE) 1985-10-23 EP disclosed
US-4540776-A Reactive fluorotriazinylaminonaphthotriazolyphenylazopyridone or pyrimidone dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1985-09-10 US disclosed
EP-0120255-A1 Reactive dyes BAYER AG (DE) 1984-10-03 EP disclosed
EP-0093306-A1 Methods for the preparation of azo compounds, and azo compounds BAYER AG (DE) 1983-11-09 EP disclosed
EP-0088930-A2 Triazole-triazinyl azo dyes BAYER AG (DE) 1983-09-21 EP disclosed
US-4354968-A Azo reactive dyestuffs having an aryl-triazinyl-aryl diazo component BAYER AKTIENGESELLSCHAFT (DE) 1982-10-19 US disclosed
EP-0013879-B1 REACTIVE DYESTUFFS, THEIR PREPARATION AND THEIR USE FOR DYEING MATERIALS CONTAINING HYDROXYL OR AMIDE GROUPS BAYER AG (DE) 1982-09-15 EP disclosed
EP-0013879-A1 Reactive dyestuffs, their preparation and their use for dyeing materials containing hydroxyl or amide groups BAYER AG (DE) 1980-08-06 EP disclosed
US-3966703-A Asymmetrical frisazo dyestuffs derived from diazotized 2,7-diamino-carbazole BAYER AKTIENGESELLSCHAFT (DT) 1976-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060069110-A1 Substituted heterocyclic compounds and methods of use MAPT, MYLK2, IAPP ADORA2A 104/4885ADORA1 370/4885ADORA3 197/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.