SCHEMBL5262869

SCHEMBL5262869

CCC(=O)Oc1c(NC(=O)Nc2ccc(S(=O)(=O)c3ccccc3)cc2)cccc1NC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 10/20 0.45
LMNA P02545 8/20 0.42
MEN1 O00255 8/20 0.42
MAPT P10636 5/20 0.42
ALDH1A1 P00352 3/20 0.41
POLB P06746 2/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPK1 P28482 2/20 0.41
GAA P10253 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
SLC16A1 P53985 1/20 0.40
CYP2C9 P11712 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NAMPT P43490 1/20 0.40
RAF1 P04049 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5261151 0.89 HTR6 (0.38) KMT2ALMNAMEN1MAPTPOLB
SCHEMBL5259783 0.85 HTT (0.39) KMT2ALMNAMEN1MAPTPOLB
SCHEMBL5262422 0.79 L3MBTL1 (0.46) KMT2ALMNAMEN1MAPTALDH1A1
SCHEMBL5260858 0.77 HTR6 (0.38) KMT2ALMNAMEN1MAPTPOLB
SCHEMBL181377 0.74 KMT2A (0.44) KMT2AMEN1MAPTALDH1A1POLB
SCHEMBL6679298 0.74 KMT2A (0.49) KMT2ALMNAMEN1MAPTALDH1A1
Hydrochloric Acid SCHEMBL28097875 0.74 KMT2A (0.44) KMT2AMEN1MAPTALDH1A1POLB
SCHEMBL4819312 0.73 POLB (0.43) KMT2ALMNAMEN1MAPTALDH1A1
SCHEMBL5261252 0.70 CA12 (0.63) CA12CA1CA2CA9
SCHEMBL5260770 0.69 ITGB1 (0.66)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383750-B1 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS ALMIRALL LAB (ES) 2007-09-26 EP claimed
EP-1383750-B1 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS ALMIRALL LAB (ES) 2007-09-26 EP disclosed
EP-1383750-A2 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS Almirall Prodesfarma, S.A. (ES) 2004-01-28 EP disclosed
WO-2002057242-A2 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS ALMIRALL PRODESFARMA, S.A. (ES) 2002-07-25 WO disclosed