SCHEMBL5260858

SCHEMBL5260858

CCC(=O)Oc1c(NCc2c(Cl)cccc2Cl)cccc1NC(=O)Nc1ccccc1S(=O)(=O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.38
ACLY P53396 2/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CXCR2 P25025 1/20 0.35
NAMPT P43490 5/20 0.35
MAPK14 Q16539 2/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
KCNQ2 O43526 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
HTT P42858 1/20 0.35
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5261151 0.87 HTR6 (0.38) HTR6ACLYNPC1RAB9ACXCR2
SCHEMBL5259278 0.78 HTR6 (0.39) HTR6ACLYNPC1RAB9ALMNA
SCHEMBL5262869 0.77 KMT2A (0.45) NPC1RAB9ANAMPTLMNAMEN1
SCHEMBL6584494 0.75 MAPK1 (0.41) NAMPTLMNAMEN1MAPTKMT2A
SCHEMBL5259783 0.74 HTT (0.39) NPC1RAB9ALMNAMEN1MAPT
SCHEMBL5259695 0.72 CA12 (0.52) MEN1KMT2AL3MBTL1POLB
SCHEMBL5260856 0.70 FPR2 (0.50) MEN1KMT2A
SCHEMBL5260861 0.70 FPR2 (0.50) MEN1KMT2A
SCHEMBL5259740 0.70 TRPV1 (0.41) NAMPTLMNAMEN1MAPTKMT2A
SCHEMBL5262422 0.67 L3MBTL1 (0.46) NPC1RAB9ALMNAMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383750-B1 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS ALMIRALL LAB (ES) 2007-09-26 EP disclosed
EP-1383750-A2 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS Almirall Prodesfarma, S.A. (ES) 2004-01-28 EP disclosed
WO-2002057242-A2 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS ALMIRALL PRODESFARMA, S.A. (ES) 2002-07-25 WO disclosed