SCHEMBL5263274

SCHEMBL5263274

C=Cc1c(Cl)ccc2ncc(OC)nc12

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 3/20 0.34
PTPN11 Q06124 7/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
KCNH2 Q12809 2/20 0.33
HTT P42858 2/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
ALDH1A1 P00352 1/20 0.31
PDE2A O00408 1/20 0.31
PDE7A Q13946 1/20 0.31
PDE10A Q9Y233 1/20 0.31
KIT P10721 1/20 0.31
NFE2L2 Q16236 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3272172 0.88 KCNH2 (0.35) KCNH2PDE2APDE7APDE10ANFE2L2
SCHEMBL14993933 0.82 CSF1R (0.33) CSF1RPDGFRBPDGFRAKCNH2HTT
SCHEMBL18544276 0.78 PDGFRB (0.36) CSF1RPTPN11PDGFRBPDGFRAKCNH2
SCHEMBL3278550 0.78 MTNR1A (0.36) HTTRAB9ANPSR1ALDH1A1NFE2L2
SCHEMBL14400283 0.78 KCNH2 (0.39) CSF1RPTPN11PDGFRBPDGFRAKCNH2
SCHEMBL3618668 0.77 CSF1R (0.35) CSF1RPTPN11PDGFRBPDGFRAKCNH2
SCHEMBL592871 0.77 KCNH2 (0.38) KCNH2
SCHEMBL1712021 0.76 RAB9A (0.39) CSF1RPDGFRBPDGFRAHTTNPC1
SCHEMBL14372223 0.75 CSF1R (0.34) CSF1RPTPN11PDGFRBPDGFRAKCNH2
SCHEMBL5747175 0.74 CCR1 (0.35) HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070244103-A1 Novel Compounds Having an Anti-Bacterial Activity MORPHOCHEM AKTIENGESELLSCHAFT FUR KOMBINATORISCHE CHEMIE (DE) 2007-10-18 US disclosed
EP-1781650-A1 NOVEL COMPOUNDS HAVING AN ANTI-BACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2007-05-09 EP disclosed
WO-2006021448-A1 NOVEL COMPOUNDS HAVING AN ANTI-BACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2006-03-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070244103-A1 Novel Compounds Having an Anti-Bacterial Activity TOP1, TOP2A, TOP2B CSF1R 2778/4885PTPN11 4460/4885PDGFRB 4424/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.