SCHEMBL5263344

SCHEMBL5263344

CC[N]c1cccc(OCCc2ccccc2)c1C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.42
ALOX5 P09917 3/20 0.42
PPARG P37231 2/20 0.42
SIRT2 Q8IXJ6 1/20 0.41
S1PR5 Q9H228 2/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
MEN1 O00255 1/20 0.39
NR1I2 O75469 1/20 0.39
LMNA P02545 1/20 0.39
CHRM2 P08172 1/20 0.39
CYP3A4 P08684 1/20 0.39
ADRA2A P08913 1/20 0.39
MAPT P10636 1/20 0.39
OPRK1 P41145 1/20 0.39
HTR2B P41595 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KMT2A Q03164 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PDE4A P27815 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4933653 0.79 NPC1 (0.49) PTGESALOX5PPARGSIRT2S1PR5
SCHEMBL5261947 0.78 CA12 (0.47) KMT2ATAAR1
SCHEMBL12095533 0.78 SIRT2 (0.45) PTGESALOX5PPARGSIRT2S1PR5
SCHEMBL5263345 0.78 SIRT2 (0.49) PTGESALOX5PPARGSIRT2CNR1
SCHEMBL4933797 0.72 SIRT2 (0.49) PTGESALOX5SIRT2CNR1CNR2
SCHEMBL12904228 0.72 KMT2A (0.60) SIRT2CNR1CNR2MEN1NR1I2
SCHEMBL3630513 0.72 SIRT2 (0.54) PPARGSIRT2CNR1CNR2MEN1
SCHEMBL27495973 0.71 ACHE (0.54) SIRT2LMNAPDE4APDE4BPDE4C
SCHEMBL28256649 0.71 PDE4A (0.50) SIRT2S1PR5MEN1NR1I2LMNA
SCHEMBL5264763 0.70 ALDH1A1 (0.39) MEN1LMNAMAPTHTR2BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740551-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105760-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed