SCHEMBL5264763

SCHEMBL5264763

CC[N]c1cccc(C)c1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
HPGD P15428 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2B P41595 1/20 0.35
PARP1 P09874 1/20 0.34
PKM P14618 1/20 0.34
F2R P25116 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
EPHB4 P54760 1/20 0.34
RAB9A P51151 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5263526 0.81 PBRM1 (0.43) ALDH1A1HPGDLMNAPARP1TDP1
SCHEMBL5261947 0.79 CA12 (0.47) ALDH1A1L3MBTL1TDP1KDM4EKMT2A
SCHEMBL311565 0.77 PARP1 (0.46) ALDH1A1HPGDL3MBTL1DRD2HTR2A
SCHEMBL2857937 0.74 GABRA1 (0.45) ALDH1A1HTTPARP1F2REPHB4
SCHEMBL3947464 0.71 TRPA1 (0.39) ALDH1A1HPGDL3MBTL1LMNAHTT
SCHEMBL442008 0.71 TSHR (0.43) ALDH1A1HPGDL3MBTL1LMNAHTT
SCHEMBL2540273 0.70 PARP1 (0.46) ALDH1A1HPGDL3MBTL1LMNAHTT
SCHEMBL30788037 0.70 THRB (0.52) ALDH1A1HPGDPARP1KDM4EMAPT
SCHEMBL3713424 0.70 THRB (0.52) ALDH1A1HPGDPARP1KDM4EMAPT
SCHEMBL689849 0.70 CD44 (0.48) ALDH1A1HPGDL3MBTL1DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740551-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105760-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed