SCHEMBL5263541

SCHEMBL5263541

C=CCc1c(C)ccc2nc(C(C(=O)O)[N+](=O)[O-])ccc12

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.34
KDM4E B2RXH2 2/20 0.31
MAPK1 P28482 1/20 0.31
GAA P10253 1/20 0.31
TSHR P16473 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
RXRA P19793 1/20 0.30
NR4A2 P43354 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5263549 1.00 ALDH1A1 (0.35) ALDH1A1MAPTKDM4EMAPK1GAA
SCHEMBL429986 0.76 ALDH1A1 (0.45) ALDH1A1MAPTKDM4EMAPK1GAA
SCHEMBL429018 0.74 ALDH1A1 (0.37) ALDH1A1KDM4EGAATSHRSMN1; SMN2
SCHEMBL429019 0.74 ALDH1A1 (0.37) ALDH1A1KDM4EGAATSHRSMN1; SMN2
SCHEMBL425787 0.73 HSD17B10 (0.39) ALDH1A1MAPTKDM4EMAPK1TSHR
SCHEMBL428060 0.64 TDP1 (0.40) ALDH1A1MAPTKDM4EMAPK1TSHR
SCHEMBL428061 0.64 TDP1 (0.40) ALDH1A1MAPTKDM4EMAPK1TSHR
SCHEMBL430744 0.62 MAPT (0.47) ALDH1A1MAPTKDM4ETSHRSMN1; SMN2
SCHEMBL426942 0.62 PTGS2 (0.42) ALDH1A1MAPTKDM4ESMN1; SMN2HSD17B10
SCHEMBL428326 0.61 GPR35 (0.42) ALDH1A1MAPTTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786822-A1 FUSED TRICYCLIC DERIVATIVES FOR THE TREATMENT OF PSYCHOTIC DISORDERS GLAXO GROUP LIMITED (GB) 2007-05-23 EP disclosed
WO-2006024517-A1 FUSED TRICYCLIC DERIVATIVES FOR THE TREATMENT OF PSYCHOTIC DISORDERS GLAXO GROUP LIMITED (GB) 2006-03-09 WO disclosed