SCHEMBL5264197

SCHEMBL5264197

COc1ccc(CCNc2ncnc3sc([N+](=O)[O-])cc23)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
GALR3 O60755 2/20 0.53
NR2F2 P24468 2/20 0.53
PDE5A O76074 1/20 0.52
AURKA O14965 1/20 0.48
RPS6KB1 P23443 1/20 0.48
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA13 Q8N1Q1 1/20 0.47
LMNA P02545 5/20 0.47
HTT P42858 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 5/20 0.46
TP53 P04637 3/20 0.46
POLB P06746 1/20 0.45
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5439670 0.82 RAB9A (0.74) NPC1RAB9AGALR3NR2F2AURKA
SCHEMBL5264803 0.81 NPC1 (0.57) NPC1RAB9AGALR3NR2F2AURKA
SCHEMBL5429336 0.81 KDM4E (0.61) NPC1RAB9AGALR3NR2F2AURKA
SCHEMBL5436053 0.80 NPC1 (0.55) NPC1RAB9AGALR3NR2F2AURKA
SCHEMBL5423720 0.80 NPC1 (0.55) NPC1RAB9AGALR3NR2F2AURKA
SCHEMBL2187106 0.78 EGFR (0.54)
SCHEMBL7465161 0.76 PDE5A (0.52) PDE5AAURKARPS6KB1LMNAHTT
SCHEMBL5423236 0.75 RAB9A (0.73) NPC1RAB9AGALR3NR2F2AURKA
SCHEMBL27697469 0.74 NPC1 (0.49) NPC1RAB9AGALR3NR2F2AURKA
SCHEMBL11414153 0.74 EGFR (0.64) RAB9AGALR3NR2F2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802632-A1 THIENO-PYRIMIDINE COMPOUNDS HAVING FUNGICIDAL ACTIVITY Dow AgroSciences LLC (US) 2007-07-04 EP disclosed
WO-2006047397-A1 THIENO-PYRIMIDINE COMPOUNDS HAVING FUNGICIDAL ACTIVITY DOW AGROSCIENCES LLC (US) 2006-05-04 WO disclosed