SCHEMBL5264362

SCHEMBL5264362

Cc1c(Cc2ccc(F)cc2)ccc2[nH]c(=O)oc(=O)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
ACHE P22303 1/20 0.46
CNR2 P34972 2/20 0.43
GPR55 Q9Y2T6 2/20 0.43
HCAR2 Q8TDS4 1/20 0.42
CNR1 P21554 1/20 0.42
AR P10275 1/20 0.38
MAPT P10636 3/20 0.36
RET P07949 1/20 0.36
KDR P35968 1/20 0.36
IL4I1 Q96RQ9 1/20 0.36
BRD4 O60885 1/20 0.36
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5263339 0.88 MAOA (0.47) MAOAMAOBACHECNR2GPR55
SCHEMBL18584304 0.82 MAOA (0.44) MAOAMAOBACHECNR2GPR55
SCHEMBL17522757 0.77 MAOA (0.45) MAOAMAOBACHECNR2GPR55
SCHEMBL17501700 0.77 MAOA (0.46) MAOAMAOBACHECNR2GPR55
SCHEMBL4492747 0.73 NOS1 (0.44) MAOAMAOBACHEARNOS1
SCHEMBL4502778 0.70 NOS1 (0.42) MAOAMAOBACHEARNOS1
SCHEMBL6508140 0.70 ESR1 (0.44) MAOAMAOBACHEARNOS1
SCHEMBL6499021 0.70 MAPT (0.43) MAPTBRD4ALDH1A1LMNAGAA
SCHEMBL15823883 0.69 CYP1A2 (0.52) MAOAMAOBGPR55IL4I1ALDH1A1
SCHEMBL6496075 0.68 NOS1 (0.40) MAOAMAOBACHEARMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786807-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2007-05-23 EP disclosed
WO-2006021340-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2006-03-02 WO disclosed