SCHEMBL5263339

SCHEMBL5263339

O=c1[nH]c2ccc(Cc3ccc(F)cc3)c(F)c2c(=O)o1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 5/20 0.47
MAOB P27338 5/20 0.47
ACHE P22303 1/20 0.47
HCAR2 Q8TDS4 1/20 0.43
CNR2 P34972 2/20 0.36
GPR55 Q9Y2T6 2/20 0.36
IL4I1 Q96RQ9 1/20 0.36
MAPT P10636 1/20 0.35
PPM1D O15297 1/20 0.35
CNR1 P21554 1/20 0.35
F2 P00734 1/20 0.34
CFD P00746 1/20 0.34
AR P10275 1/20 0.34
GRIN2D O15399 2/20 0.33
GRIN3B O60391 2/20 0.33
GRIN1 Q05586 2/20 0.33
GRIN2A Q12879 2/20 0.33
GRIN2B Q13224 2/20 0.33
GRIN2C Q14957 2/20 0.33
GRIN3A Q8TCU5 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5264362 0.88 MAOA (0.46) MAOAMAOBACHEHCAR2CNR2
SCHEMBL18584304 0.83 MAOA (0.44) MAOAMAOBACHEHCAR2CNR2
SCHEMBL17522757 0.78 MAOA (0.45) MAOAMAOBACHEHCAR2CNR2
SCHEMBL17501700 0.76 MAOA (0.46) MAOAMAOBACHECNR2GPR55
SCHEMBL537909 0.74 F2 (0.43) MAOAMAOBACHEF2CFD
SCHEMBL4502778 0.71 NOS1 (0.42) MAOAMAOBACHEF2CFD
SCHEMBL15823883 0.70 CYP1A2 (0.52) MAOAMAOBGPR55IL4I1F2
SCHEMBL10343102 0.66 F2 (0.50) MAOAMAOBIL4I1F2CFD
SCHEMBL3576862 0.65 NOS1 (0.42) MAOAMAOBACHEF2CFD
SCHEMBL694149 0.64 MAOA (0.61) MAOAMAOBACHEF2CFD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786807-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2007-05-23 EP disclosed
WO-2006021340-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2006-03-02 WO disclosed