SCHEMBL5264458

SCHEMBL5264458

COC(=O)C(Cc1ccc(OC(=O)N2CCN(C)CC2)cc1)NC(=O)Nc1ccccc1S(=O)(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.51
ITGA4 P13612 1/20 0.51
ITGB7 P26010 1/20 0.51
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
YAP1 P46937 1/20 0.43
NLRP3 Q96P20 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
POLB P06746 1/20 0.42
GFER P55789 1/20 0.42
CACNA1B Q00975 1/20 0.41
CTSB P07858 2/20 0.41
P2RX7 Q99572 6/20 0.41
ATM Q13315 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5264453 1.00 ITGB1 (0.51) ITGB1ITGA4ITGB7CA12CA1
SCHEMBL6642120 0.98 ITGB1 (0.55) ITGB1ITGA4ITGB7CA12CA1
SCHEMBL5265251 0.93 ITGB1 (0.59) ITGB1ITGA4ITGB7YAP1CTSB
SCHEMBL5265258 0.93 ITGB1 (0.59) ITGB1ITGA4ITGB7YAP1CTSB
SCHEMBL5261098 0.83 CA12 (0.49) ITGB1ITGA4CA12CA1CA2
SCHEMBL5262420 0.83 CA12 (0.49) ITGB1ITGA4CA12CA1CA2
SCHEMBL5258179 0.81 CA12 (0.55) CA12CA1CA2CA9NLRP3
SCHEMBL5258183 0.81 CA12 (0.55) CA12CA1CA2CA9NLRP3
SCHEMBL5260154 0.80 CA12 (0.57) CA12CA1CA2CA9NLRP3
SCHEMBL5260159 0.80 CA12 (0.57) CA12CA1CA2CA9NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383750-B1 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS ALMIRALL LAB (ES) 2007-09-26 EP claimed
US-7253171-B2 Urea derivatives as integrin α4 antagonists LABORATORIOS ALMIRALL, S.A. (ES) 2007-08-07 US claimed
US-20040142982-A1 Urea derivatives as integrin alpha 4 antagonists LABORATORIOS ALMIRALL, S.A. (ES) 2004-07-22 US claimed
US-20070238763-A1 Urea derivatives as integrin a4 antagonists LABORATORIOS ALMIRALL, S.A. 2007-10-11 US disclosed
EP-1383750-B1 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS ALMIRALL LAB (ES) 2007-09-26 EP disclosed
US-7253171-B2 Urea derivatives as integrin α4 antagonists LABORATORIOS ALMIRALL, S.A. (ES) 2007-08-07 US disclosed
US-20040142982-A1 Urea derivatives as integrin alpha 4 antagonists LABORATORIOS ALMIRALL, S.A. (ES) 2004-07-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040142982-A1 Urea derivatives as integrin alpha 4 antagonists ITGA4, ITGB4, ITGA1 ITGB1 4/4885ITGA4 1/4885ITGB7 14/4885
US-20070238763-A1 Urea derivatives as integrin a4 antagonists ITGB4, ITGA4, ITGB7 ITGB1 5/4885ITGA4 2/4885ITGB7 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.