SCHEMBL5264564

SCHEMBL5264564

Cc1ccc(S(=O)(=O)n2ccc3c(CC=O)ncnc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.50
RAPGEF4 Q8WZA2 2/20 0.39
KDM4E B2RXH2 1/20 0.39
UBE2N P61088 1/20 0.39
BRD4 O60885 1/20 0.38
POLB P06746 1/20 0.38
ALDH3A1 P30838 1/20 0.38
HTT P42858 1/20 0.38
NOD1 Q9Y239 1/20 0.38
HTR6 P50406 2/20 0.37
CYP19A1 P11511 1/20 0.36
PKM P14618 2/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13494114 0.86 L3MBTL1 (0.50) L3MBTL1RAPGEF4BRD4POLBALDH3A1
SCHEMBL29247903 0.82 PTGDR2 (0.47) L3MBTL1RAPGEF4KDM4EPOLBALDH3A1
SCHEMBL260617 0.80 L3MBTL1 (0.55) L3MBTL1RAPGEF4KDM4EUBE2NBRD4
SCHEMBL6726762 0.79 L3MBTL1 (0.44) L3MBTL1RAPGEF4BRD4POLBALDH3A1
SCHEMBL24262373 0.78 L3MBTL1 (0.43) L3MBTL1RAPGEF4KDM4EPOLBHTT
SCHEMBL30575111 0.78 L3MBTL1 (0.43) L3MBTL1RAPGEF4KDM4EPOLBHTT
SCHEMBL14427677 0.78 L3MBTL1 (0.52) L3MBTL1RAPGEF4KDM4EUBE2NBRD4
SCHEMBL1356181 0.78 L3MBTL1 (0.52) L3MBTL1RAPGEF4KDM4EUBE2NBRD4
SCHEMBL4075074 0.78 L3MBTL1 (0.52) L3MBTL1RAPGEF4KDM4EUBE2NBRD4
SCHEMBL28622254 0.78 L3MBTL1 (0.52) L3MBTL1RAPGEF4BRD4POLBALDH3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844050-A1 PYRROLOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASE Vertex Pharmaceuticals, Inc. (US) 2007-10-17 EP disclosed
WO-2006096270-A1 PYRROLOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-09-14 WO disclosed