SCHEMBL5264641

SCHEMBL5264641

O=CCc1cc(F)ccc1N1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.47
HTR1A P08908 10/20 0.46
SLC6A2 P23975 6/20 0.46
SLC6A4 P31645 6/20 0.46
HTR7 P34969 3/20 0.42
HTR6 P50406 5/20 0.41
SLC6A3 Q01959 3/20 0.40
HTR2B P41595 2/20 0.40
HTR3A P46098 2/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6027239 0.88 KDR (0.47) KDRHTR1ASLC6A2SLC6A4HTR7
SCHEMBL24760628 0.80 HTR1A (0.49) KDRHTR1ASLC6A2SLC6A4HTR7
SCHEMBL27474954 0.80 HTR1A (0.49) KDRHTR1ASLC6A2SLC6A4HTR7
SCHEMBL28775480 0.79 KDR (0.47) KDRHTR1ASLC6A2SLC6A4HTR7
Hydrochloric Acid SCHEMBL27621259 0.79 HTR1A (0.48) KDRHTR1ASLC6A2SLC6A4HTR7
SCHEMBL5023862 0.78 ALDH1A1 (0.45) KDRHTR1ASLC6A2SLC6A4HTR6
Tert-Butyl Formate SCHEMBL27621184 0.76 HTR1A (0.41) KDRHTR1ASLC6A2SLC6A4HTR6
Hydrochloric Acid SCHEMBL5913628 0.76 KDR (0.49) KDRHTR1ASLC6A2SLC6A4HTR7
SCHEMBL13862081 0.74 CHRNB2 (0.46) HTR1ASLC6A2SLC6A4HTR7SLC6A3
SCHEMBL233938 0.74 KDR (0.53) KDRHTR1ASLC6A2SLC6A4HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833800-A1 PYRAZOLONE COMPOUNDS AS METABOTROPIC GLUTAMATE RECEPTOR AGONISTS FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS AstraZeneca AB (SE) 2007-09-19 EP disclosed
WO-2006071730-A1 PYRAZOLONE COMPOUNDS AS METABOTROPIC GLUTAMATE RECEPTOR AGONISTS FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS ASTRAZENECA AB (SE) 2006-07-06 WO disclosed