SCHEMBL5265141

SCHEMBL5265141

CC(NC(=O)c1nc2ccccc2[nH]1)C(Cc1ccc(Cl)cc1)c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 13/20 0.49
CNR2 P34972 11/20 0.49
FAAH O00519 1/20 0.48
FDFT1 P37268 2/20 0.48
FFAR2 O15552 1/20 0.47
KMT2A Q03164 1/20 0.47
KDM4E B2RXH2 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5259431 0.86 CNR1 (0.50) CNR1CNR2FDFT1
SCHEMBL6325773 0.86 CNR1 (0.50) CNR1CNR2FDFT1
SCHEMBL5318869 0.80 CNR1 (0.48) CNR1CNR2FDFT1
SCHEMBL5265142 0.79 FAAH (0.50) CNR2FAAHFFAR2KMT2AKDM4E
SCHEMBL5262773 0.78 CNR1 (0.72) CNR1CNR2FDFT1
SCHEMBL5263205 0.77 ALOX15 (0.57) CNR1CNR2FDFT1FFAR2KMT2A
SCHEMBL5261127 0.77 CNR1 (0.49) CNR1CNR2FDFT1KDM4E
SCHEMBL5262269 0.77 CNR1 (0.63) CNR1CNR2FDFT1KMT2ARAB9A
SCHEMBL5263456 0.76 CNR1 (0.49) CNR1CNR2FDFT1
SCHEMBL5261540 0.76 CNR1 (0.60) CNR1CNR2FDFT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP claimed
JP-2005527586-A 2005-09-15 JP claimed
US-20050154202-A1 Substituted aryl amides MERCK & CO., INC. 2005-07-14 US claimed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP claimed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO claimed
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP disclosed
US-20050154202-A1 Substituted aryl amides MERCK & CO., INC. 2005-07-14 US disclosed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP disclosed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050154202-A1 Substituted aryl amides CNR1, CNR2, FAAH CNR1 1/4885CNR2 2/4885FAAH 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.