SCHEMBL5265142

SCHEMBL5265142

CC(c1ccc(Cl)cc1)C(CNC(=O)c1nc2ccccc2[nH]1)c1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.50
FFAR2 O15552 1/20 0.49
NPC1 O15118 6/20 0.47
RAB9A P51151 6/20 0.47
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
MAPT P10636 5/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
LMNA P02545 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
ALDH1A1 P00352 3/20 0.45
HTT P42858 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5259433 0.85 HRH4 (0.42) FAAHFFAR2RAB9AMEN1KMT2A
SCHEMBL5265141 0.79 CNR1 (0.49) FAAHFFAR2NPC1RAB9AKMT2A
SCHEMBL5262774 0.77 SLC6A9 (0.54) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL5262685 0.76 KDM4E (0.47) FAAHFFAR2MAPTLMNASMN1; SMN2
SCHEMBL5264318 0.76 ALOX15 (0.56) FFAR2NPC1RAB9AHDAC3HDAC1
SCHEMBL5266049 0.76 RAB9A (0.60) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL5263458 0.75 L3MBTL1 (0.42) FFAR2NPC1RAB9AMAPTMEN1
SCHEMBL5261544 0.75 TLR7 (0.52) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL5261739 0.74 NPC1 (0.61) NPC1RAB9AALDH1A1CYP1A2HPGD
SCHEMBL5262900 0.74 NSD2 (0.45) MEN1KMT2ALMNASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP claimed
JP-2005527586-A 2005-09-15 JP claimed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP claimed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO claimed
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP disclosed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP disclosed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO disclosed