SCHEMBL5266355

SCHEMBL5266355

COC(=O)OC1CCNC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 2/20 0.35
TOP2A P11388 2/20 0.35
SLC6A1 P30531 2/20 0.34
GABRA5 P31644 2/20 0.34
GABRB2 P47870 2/20 0.34
SLC6A12 P48065 2/20 0.34
SLC6A11 P48066 2/20 0.34
SLC6A13 Q9NSD5 2/20 0.34
GABRA1 P14867 1/20 0.34
GABRR1 P24046 1/20 0.34
GABRA4 P48169 1/20 0.34
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
EPHX1 P07099 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13600289 1.00 HSP90AB1 (0.35) HSP90AB1TOP2ASLC6A1GABRA5GABRB2
SCHEMBL13600285 1.00 HSP90AB1 (0.35) HSP90AB1TOP2ASLC6A1GABRA5GABRB2
SCHEMBL2334130 0.88 EPHX1 (0.40) HSP90AB1TOP2AGABRA5GABRB2GABRA1
Hydrochloric Acid SCHEMBL10868234 0.87 SLC6A1 (0.40) SLC6A1SLC6A11SLC6A13CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL5209870 0.86 EPHX1 (0.39) HSP90AB1TOP2AGABRA5GABRB2GABRA1
SCHEMBL5155633 0.83
Hydrochloric Acid SCHEMBL7258085 0.81 CHRNB2 (0.41) CHRNB2CHRNA4EPHX1CHRNB4CHRNA3
SCHEMBL701944 0.79 ALDH1A1 (0.41) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL435813 0.79
SCHEMBL6181576 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836180-B1 SULFONYL PYRROLIDINES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS DRUGS SANOFI SA (FR) 2012-06-13 EP disclosed
EP-1836180-A2 SULFONYL PYRROLIDINES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS DRUGS sanofi-aventis (FR) 2007-09-26 EP disclosed
WO-2006072393-A2 SULFONYL PYRROLIDINES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS DRUGS SANOFI-AVENTIS (DE) 2006-07-13 WO disclosed