SCHEMBL5269941

SCHEMBL5269941

O=C(Nc1c[nH]nc1C(=O)NCc1ccccc1)c1ccc2[nH]ccc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFATC1 O95644 1/20 0.47
PADI4 Q9UM07 1/20 0.47
PADI2 Q9Y2J8 1/20 0.47
NR1H4 Q96RI1 1/20 0.46
NPC1 O15118 1/20 0.46
MAPT P10636 1/20 0.46
RAB9A P51151 1/20 0.46
ROCK1 Q13464 2/20 0.45
JAK2 O60674 1/20 0.45
MAP4K4 O95819 1/20 0.45
CHEK2 O96017 1/20 0.45
PRKCG P05129 1/20 0.45
CDK1 P06493 1/20 0.45
FES P07332 1/20 0.45
RET P07949 1/20 0.45
ROS1 P08922 1/20 0.45
FER P16591 1/20 0.45
FLT1 P17948 1/20 0.45
AXL P30530 1/20 0.45
FLT4 P35916 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5269216 0.90 HDAC1 (0.46) NFATC1PADI4PADI2NPC1MAPT
SCHEMBL5267173 0.85 HPGD (0.49) NPC1MAPTRAB9A
SCHEMBL5274230 0.83 HPGD (0.49) ROCK1MAP4K4PRKCGPKN2MAP4K5
SCHEMBL9764513 0.82 CTNNB1 (0.58) NFATC1PADI4PADI2NR1H4NPC1
SCHEMBL5269714 0.81 ROCK2 (0.54) NR1H4NPC1RAB9AROCK1MAP4K4
SCHEMBL5265277 0.80 TAS1R3 (0.50) NFATC1NPC1MAPTRAB9AMAOA
SCHEMBL5269031 0.79 HPGD (0.62) HDAC1MAPK14
SCHEMBL5320217 0.78 MAPK14 (0.55) NR1H4RAB9AROCK1MAP4K4PRKCG
SCHEMBL5270246 0.78 NPC1 (0.57) NPC1MAPTRAB9AHDAC3HDAC1
SCHEMBL5271804 0.77 SMYD3 (0.51) NPC1MAPTRAB9AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed