SCHEMBL5272020

SCHEMBL5272020

CC(=O)c1ccc2c(c1)N(C(=O)CN1CCc3ccccc3C1C)c1ccccc1S2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 2/20 0.48
MAPT P10636 3/20 0.47
LMNA P02545 3/20 0.47
MAPK1 P28482 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP2D6 P10635 4/20 0.46
CYP1A2 P05177 3/20 0.46
CYP3A4 P08684 2/20 0.46
TSHR P16473 2/20 0.46
CYP2C19 P33261 1/20 0.46
ALDH1A1 P00352 3/20 0.45
USP2 O75604 2/20 0.44
ALOX15 P16050 1/20 0.44
HTR1A P08908 3/20 0.43
DRD2 P14416 3/20 0.43
SLC6A2 P23975 3/20 0.43
SLC6A4 P31645 3/20 0.43
ADRA1A P35348 3/20 0.43
DRD3 P35462 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5241937 0.88 BCHE (0.44) NOX1MAPTLMNAMAPK1TDP1
SCHEMBL5243732 0.86 CYP3A4 (0.46) MAPTLMNAMAPK1TDP1CYP2D6
SCHEMBL5243083 0.78 KMT2A (0.49) CYP2D6CYP1A2CYP3A4TSHRCYP2C19
SCHEMBL5468076 0.76 CYP3A4 (0.48) NOX1MAPTLMNAMAPK1TDP1
SCHEMBL5280780 0.76 BCHE (0.52) MAPTLMNACYP2D6CYP1A2CYP3A4
SCHEMBL5278993 0.75 BCHE (0.45) NOX1MAPTLMNAMAPK1TDP1
SCHEMBL5456545 0.74 CYP3A4 (0.48) NOX1MAPTLMNAMAPK1TDP1
SCHEMBL5467983 0.74 CYP3A4 (0.48) NOX1MAPTLMNAMAPK1TDP1
SCHEMBL5350976 0.74 KMT2A (0.55) LMNACYP1A2CYP3A4TSHRCYP2C19
SCHEMBL30725912 0.72 NOX1 (0.73) NOX1MAPTLMNAMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833797-A1 AZACYCLIC COMPOUNDS AS INHBITORS OF SENSORY NEURONE SPECIFIC CHANNELS (SNS) VERNALIS (R&D) LTD (GB) 2007-09-19 EP disclosed
WO-2006082354-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS ( SNS ) VERNALIS (R & D) LIMITED (GB) 2006-08-10 WO disclosed