SCHEMBL5243083

SCHEMBL5243083

COc1cc2c(cc1OC)C(C)N(CC(=O)N1c3ccccc3Sc3ccccc31)CC2

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
NPC1 O15118 1/20 0.48
POLB P06746 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
HCRTR1 O43613 5/20 0.47
HCRTR2 O43614 4/20 0.47
ALDH1A1 P00352 2/20 0.47
USP2 O75604 1/20 0.46
ALOX15 P16050 1/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP1A2 P05177 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5280780 0.93 BCHE (0.52) KMT2AALDH1A1CYP3A4CYP2D6CYP1A2
SCHEMBL5241937 0.92 BCHE (0.44) KMT2ANPC1POLBSMN1; SMN2HCRTR1
SCHEMBL5350976 0.91 KMT2A (0.55) KMT2AALDH1A1CYP3A4CYP1A2TSHR
SCHEMBL5243272 0.86 SMN1; SMN2 (0.52) KMT2ANPC1POLBSMN1; SMN2HCRTR1
SCHEMBL5334834 0.82 SMN1; SMN2 (0.59) KMT2ANPC1POLBSMN1; SMN2ALDH1A1
SCHEMBL5241484 0.80 BCHE (0.47) KMT2ASMN1; SMN2ALDH1A1USP2ALOX15
SCHEMBL5466400 0.79 ALDH1A1 (0.56) KMT2APOLBSMN1; SMN2ALDH1A1USP2
SCHEMBL5272020 0.78 NOX1 (0.48) KMT2AALDH1A1USP2ALOX15CYP3A4
SCHEMBL5243732 0.77 CYP3A4 (0.46) KMT2ANPC1SMN1; SMN2ALDH1A1USP2
SCHEMBL5289084 0.77 SMN1; SMN2 (0.61) KMT2ANPC1POLBSMN1; SMN2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833797-A1 AZACYCLIC COMPOUNDS AS INHBITORS OF SENSORY NEURONE SPECIFIC CHANNELS (SNS) VERNALIS (R&D) LTD (GB) 2007-09-19 EP disclosed
WO-2006082354-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS ( SNS ) VERNALIS (R & D) LIMITED (GB) 2006-08-10 WO disclosed