SCHEMBL527216

SCHEMBL527216

Clc1cc2cc3c(cc2nn1)OCO3

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
HSD17B10 Q99714 6/20 0.40
KDM4E B2RXH2 5/20 0.40
HPGD P15428 5/20 0.40
MAPT P10636 4/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
TP53 P04637 3/20 0.40
TSHR P16473 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
PKM P14618 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
SRC P12931 1/20 0.38
RPS6KB2 Q9UBS0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5562603 0.74 SRC (0.42) ALDH1A1HSD17B10KDM4EHPGDMAPT
SCHEMBL527950 0.73 KDM4E (0.43) ALDH1A1HSD17B10KDM4EHPGDMAPT
SCHEMBL1650792 0.73 ALDH1A1 (0.43) ALDH1A1HSD17B10KDM4EHPGDMAPT
SCHEMBL30250019 0.67 CYP3A4 (0.57) ALDH1A1HSD17B10KDM4EHPGDMAPT
SCHEMBL10638685 0.67 ALDH1A1 (0.57) ALDH1A1HSD17B10KDM4EHPGDMAPT
SCHEMBL10635467 0.67 CYP3A4 (0.57) ALDH1A1HSD17B10KDM4EHPGDMAPT
SCHEMBL2359770 0.67 PDGFRB (0.41) ALDH1A1HSD17B10KDM4EHPGDMAPT
SCHEMBL13993586 0.67 MPO (0.40) ALDH1A1HSD17B10KDM4EHPGDMAPT
SCHEMBL241448 0.67 MPO (0.40) ALDH1A1HSD17B10KDM4EHPGDMAPT
SCHEMBL3783578 0.67 EGFR (0.44) ALDH1A1HSD17B10KDM4EHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012015901-A1 METHODS FOR TREATING GASTRIC AND PANCREATIC MALIGNANCIES GENZYME CORPORATION (US) 2012-02-02 WO disclosed