SCHEMBL5274263

SCHEMBL5274263

O=C(NCc1ccc(Cl)cc1Cl)Oc1cn(C2CC2)c2c(Cl)c(N3CCCN(CCO)CC3)c(F)cc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
P2RX7 Q99572 7/20 0.37
EPHX2 P34913 3/20 0.37
MAPK8 P45983 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5282397 0.91 ALDH1A1 (0.40) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL968075 0.90 ALDH1A1 (0.45) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5164103 0.87 ALDH1A1 (0.43) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5284805 0.85 ALDH1A1 (0.39) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5279472 0.84 ALDH1A1 (0.50) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5279342 0.83 EPHX2 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5280454 0.83 EPHX2 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5280465 0.83 EPHX2 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5178320 0.83 KDM4E (0.36) ALDH1A1POLBOPRM1P2RX7EPHX2
SCHEMBL5283636 0.83 POLB (0.43) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768973-B1 SUBSTITUTED QUINOLONES AICURIS GMBH & CO KG (DE) 2007-12-05 EP disclosed