SCHEMBL5275098

SCHEMBL5275098

Cc1scc(NC(=O)CCc2ccc(-c3ccccc3)cc2)c1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 18/20 0.56
LTB4R Q15722 1/20 0.53
POLB P06746 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3552606 0.82 MMP3 (0.57)
SCHEMBL13781563 0.81 HCAR2 (0.52) HCAR2LTB4RPOLB
SCHEMBL3561642 0.80 SLC12A2 (0.41) HCAR2POLB
SCHEMBL3561743 0.80 NPC1 (0.55) HCAR2POLB
SCHEMBL13781560 0.78 ALDH1A1 (0.56) HCAR2LTB4RPOLB
SCHEMBL12756640 0.77 HCAR2 (0.59) HCAR2
SCHEMBL1490241 0.76 ALOX15 (0.53) HCAR2
SCHEMBL1490744 0.76 HDAC2 (0.47) HCAR2POLB
SCHEMBL1490571 0.76 HCAR2 (0.59) HCAR2POLB
SCHEMBL5062205 0.76 HCAR2 (0.64) HCAR2LTB4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1853579-A2 2-SUBSTITUTED 5-MEMBERED HETEROARYL CARBOXYLATES AS HM74A RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-11-14 EP disclosed
WO-2006085113-A2 2-SUBSTITUTED 5-MEMBERED HETEROARYL CARBOXYLATES AS HM74A RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2006-08-17 WO disclosed