SCHEMBL5278014

SCHEMBL5278014

CCC(CC)N[C@@H]1COc2ccc(C(=O)O)cc2C1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.48
TAS1R3 Q7RTX0 3/20 0.44
TAS1R1 Q7RTX1 3/20 0.44
MTNR1A P48039 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.41
ROCK2 O75116 1/20 0.41
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
HCAR3 P49019 1/20 0.38
MAPT P10636 1/20 0.37
RARA P10276 1/20 0.37
RARB P10826 1/20 0.37
RARG P13631 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
HDAC8 Q9BY41 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9441687 0.74 DRD3 (0.57) TDP1
Hydrochloric Acid SCHEMBL9441693 0.73 DRD3 (0.56) TDP1
SCHEMBL5238494 0.72 MTNR1A (0.45) TDP1TAS1R3TAS1R1MTNR1AMAPT
SCHEMBL5278012 0.72 DRD3 (0.55) TDP1
SCHEMBL5237994 0.72 DRD3 (0.55) TDP1
SCHEMBL25959765 0.72 ROCK2 (0.53) TDP1MTNR1AROCK2ALDH1A1MAPK1
SCHEMBL27927241 0.72 TDP1 (0.55) TDP1ROCK2ALDH1A1MAPK1RARA
SCHEMBL5241204 0.71 MTNR1A (0.44) TAS1R3TAS1R1MTNR1AMAPTITGB3
SCHEMBL5238670 0.69 MTNR1A (0.42) TAS1R3TAS1R1MTNR1AMAPTITGB3
SCHEMBL5238113 0.68 DRD3 (0.51) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1819690-A2 CHROMAN COMPOUNDS Pfizer Limited (GB) 2007-08-22 EP disclosed
WO-2006056850-A2 CHROMAN COMPOUNDS PFIZER LIMITED (GB) 2006-06-01 WO disclosed