SCHEMBL5280063

SCHEMBL5280063

CCOC(=O)Oc1cnc(-c2ccccc2)nc1Oc1ccccc1C#N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.49
CYP2C9 P11712 4/20 0.49
CYP2C19 P33261 4/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
POLB P06746 2/20 0.49
ALDH1A1 P00352 8/20 0.46
LMNA P02545 2/20 0.46
NPSR1 Q6W5P4 4/20 0.46
KDM4E B2RXH2 2/20 0.46
CYP3A4 P08684 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
MAPT P10636 3/20 0.45
MAPK1 P28482 1/20 0.45
ATM Q13315 1/20 0.45
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
NPC1 O15118 1/20 0.44
TP53 P04637 1/20 0.44
RAB9A P51151 1/20 0.44
GPR55 Q9Y2T6 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5280353 0.87 ALDH1A1 (0.49) CYP1A2CYP2C9CYP2C19L3MBTL1POLB
SCHEMBL5282395 0.86 ALDH1A1 (0.64) CYP1A2CYP2C9CYP2C19L3MBTL1POLB
SCHEMBL5124969 0.84 CYP1A2 (0.71) CYP1A2CYP2C9CYP2C19L3MBTL1POLB
SCHEMBL5279716 0.84 CYP1A2 (0.46) CYP1A2CYP2C9CYP2C19L3MBTL1POLB
SCHEMBL5286570 0.83 NPSR1 (0.66) CYP1A2CYP2C9CYP2C19L3MBTL1POLB
SCHEMBL5279673 0.80 ALDH1A1 (0.50) CYP1A2CYP2C9CYP2C19L3MBTL1POLB
SCHEMBL5280788 0.80 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19L3MBTL1POLB
SCHEMBL5124890 0.79 KMT2A (0.64) CYP1A2CYP2C9CYP2C19L3MBTL1POLB
SCHEMBL5282772 0.78 L3MBTL1 (0.56) CYP1A2CYP2C9CYP2C19L3MBTL1POLB
SCHEMBL3658119 0.78 ALDH1A1 (0.51) L3MBTL1POLBALDH1A1NPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866289-A1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES AND USE THEREOF Bayer HealthCare AG (DE) 2007-12-19 EP disclosed
WO-2006097220-A1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES AND USE THEREOF BAYER HEALTHCARE AG (DE) 2006-09-21 WO disclosed