SCHEMBL5280353

SCHEMBL5280353

N#Cc1ccccc1Oc1nc(-c2ccccc2)ncc1OC(=O)O

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
PIN1 Q13526 2/20 0.47
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
NPSR1 Q6W5P4 3/20 0.46
CYP1A2 P05177 4/20 0.42
CYP2C9 P11712 4/20 0.42
CYP2C19 P33261 4/20 0.42
MAPT P10636 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
CYP3A4 P08684 2/20 0.40
MAPK14 Q16539 1/20 0.39
LMNA P02545 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5280063 0.87 CYP1A2 (0.49) ALDH1A1PIN1KMT2AMEN1NPSR1
SCHEMBL5124890 0.84 KMT2A (0.64) ALDH1A1PIN1KMT2AMEN1CYP1A2
SCHEMBL5279608 0.83 ALDH1A1 (0.71) ALDH1A1KMT2AMEN1NPSR1CYP1A2
SCHEMBL5285487 0.81 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1NPSR1CYP1A2
SCHEMBL5284020 0.81 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1NPSR1CYP1A2
SCHEMBL5294553 0.81 ALDH1A1 (0.50) ALDH1A1KMT2AMEN1NPSR1CYP1A2
SCHEMBL5279202 0.80 KMT2A (0.73) ALDH1A1KMT2AMEN1NPSR1CYP1A2
SCHEMBL5124969 0.79 CYP1A2 (0.71) ALDH1A1KMT2AMEN1NPSR1CYP1A2
SCHEMBL5279902 0.79 KMT2A (0.49) ALDH1A1KMT2AMEN1NPSR1CYP1A2
SCHEMBL14746303 0.79 PIN1 (0.43) ALDH1A1PIN1KMT2AMEN1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866289-A1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES AND USE THEREOF Bayer HealthCare AG (DE) 2007-12-19 EP disclosed
WO-2006097220-A1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES AND USE THEREOF BAYER HEALTHCARE AG (DE) 2006-09-21 WO disclosed