SCHEMBL5280227

SCHEMBL5280227

COc1ccc2c(CCN3CCC(CCNC(=O)COCc4ccc(F)cc4)CC3)c[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.49
BCHE P06276 5/20 0.49
MTNR1A P48039 1/20 0.45
MTNR1B P49286 1/20 0.45
HTR1A P08908 1/20 0.45
SLC6A4 P31645 1/20 0.45
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
CCR3 P51677 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5287676 0.94 ACHE (0.57) ACHEBCHEMTNR1AMTNR1BHTR1A
SCHEMBL6038046 0.91 ACHE (0.48) ACHEBCHEMTNR1AMTNR1B
SCHEMBL5278655 0.88 BCHE (0.59) ACHEBCHE
SCHEMBL6037985 0.85 BCHE (0.55) ACHEBCHEMTNR1AMTNR1B
SCHEMBL5279913 0.83 BCHE (0.60) ACHEBCHEHTR1ASLC6A4
SCHEMBL5281968 0.79 SPR (0.54) ACHEBCHEMTNR1AMTNR1BHTR1A
SCHEMBL5282166 0.79 ACHE (0.53) ACHEBCHEHTR1A
SCHEMBL5282667 0.77 BCHE (0.55) ACHEBCHE
SCHEMBL5291489 0.76 BCHE (0.52) ACHEBCHE
SCHEMBL5289480 0.75 BCHE (0.56) ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863804-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2007-12-12 EP claimed
WO-2006102760-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2006-10-05 WO claimed