SCHEMBL5281014

SCHEMBL5281014

NC(=O)COCc1ccc(F)c(CCCc2ccc(CN3CCC(c4c[nH]c5ccccc45)CC3)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
OPRM1 P35372 2/20 0.45
OPRK1 P41145 2/20 0.45
OPRL1 P41146 2/20 0.45
CHRM4 P08173 1/20 0.45
SLC6A4 P31645 1/20 0.44
CCR2 P41597 4/20 0.43
ADRA1D P25100 3/20 0.41
KMT2A Q03164 1/20 0.41
HTR1D P28221 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5280164 0.79 BCHE (0.43) SLC6A4KMT2A
SCHEMBL6038004 0.78 CCR2 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5340262 0.71 HDAC3 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6785509 0.71 HDAC1 (0.67) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9032088 0.70 OPRM1 (0.75) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3380970 0.69 SLC6A4 (0.71) SLC6A4CCR2ADRA1D
SCHEMBL6783190 0.67 CHRM4 (0.60) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28800093 0.67 KDM4E (0.69) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7092859 0.66 HRH2 (0.61) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6705926 0.66 CHRM4 (0.73) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863804-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2007-12-12 EP claimed
WO-2006102760-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2006-10-05 WO claimed