SCHEMBL5280164

SCHEMBL5280164

NC(=O)COCc1ccc(F)c(CCCCC2CCN(Cc3c[nH]c4ccccc34)C2)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BCHE P06276 7/20 0.43
ACHE P22303 6/20 0.43
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
SOS1 Q07889 3/20 0.42
DRD2 P14416 1/20 0.42
CYP2D6 P10635 1/20 0.40
HTR1A P08908 1/20 0.40
SLC6A4 P31645 1/20 0.40
NPC1 O15118 1/20 0.39
KRAS P01116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5279974 0.81 ALDH1A1 (0.40) BCHEACHEALDH1A1MEN1MAPK1
SCHEMBL5281014 0.79 HDAC3 (0.49) KMT2ASLC6A4
SCHEMBL5291953 0.79 BCHE (0.44) BCHEACHEALDH1A1HTR1A
SCHEMBL5279163 0.79 BCHE (0.50) BCHEACHEALDH1A1MEN1MAPK1
SCHEMBL5283383 0.76 ACHE (0.41) BCHEACHEMEN1KMT2AHTR1A
SCHEMBL5276908 0.73 TACR1 (0.36) MEN1KMT2ANPC1
SCHEMBL5279913 0.68 BCHE (0.60) BCHEACHEDRD2HTR1ASLC6A4
SCHEMBL5277140 0.67 CCR1 (0.45) BCHEACHEALDH1A1MEN1MAPK1
SCHEMBL6038039 0.67 CCR1 (0.45) BCHEACHEALDH1A1MEN1MAPK1
SCHEMBL5277138 0.67 CCR1 (0.45) BCHEACHEALDH1A1MEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863804-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2007-12-12 EP claimed
WO-2006102760-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2006-10-05 WO claimed