SCHEMBL5281269

SCHEMBL5281269

CCOC(=O)Oc1cnc(-c2ccc(C)c(C)c2)nc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
KDM4E B2RXH2 3/20 0.41
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
MAPT P10636 4/20 0.39
LMNA P02545 3/20 0.39
MAPK1 P28482 1/20 0.39
ATM Q13315 1/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
TP53 P04637 3/20 0.39
CYP1A2 P05177 4/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
POLB P06746 2/20 0.38
HSD17B10 Q99714 1/20 0.38
CUL4A Q13619 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5278782 0.92 CYP1A2 (0.42) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA
SCHEMBL5278083 0.90 ALDH1A1 (0.39) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA
SCHEMBL5282908 0.87 S1PR1 (0.41) ALDH1A1KDM4ES1PR1S1PR3SMN1; SMN2
SCHEMBL5279567 0.84 ALDH1A1 (0.56) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA
SCHEMBL5280720 0.83 PDGFRB (0.42) ALDH1A1KDM4EATMNPC1CYP1A2
SCHEMBL5111120 0.83 ALDH1A1 (0.60) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA
SCHEMBL5296815 0.83 MAPT (0.48) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL5292147 0.82 CYP11B2 (0.41) ALDH1A1KDM4EMAPTHSD17B10L3MBTL1
SCHEMBL5298454 0.81 CYP1A2 (0.39) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA
SCHEMBL5283181 0.81 ALDH1A1 (0.39) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866289-A1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES AND USE THEREOF Bayer HealthCare AG (DE) 2007-12-19 EP disclosed
WO-2006097220-A1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES AND USE THEREOF BAYER HEALTHCARE AG (DE) 2006-09-21 WO disclosed