SCHEMBL5281573

SCHEMBL5281573

CCOC(=O)C(C#N)c1ccc2ccccc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
SLC6A2 P23975 2/20 0.45
SLC6A4 P31645 2/20 0.45
SLC6A3 Q01959 2/20 0.45
CYP2D6 P10635 1/20 0.45
KCNH2 Q12809 1/20 0.45
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
UGT2B7 P16662 1/20 0.42
GLA P06280 1/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41
TSHR P16473 1/20 0.41
CASP1 P29466 1/20 0.41
MMP13 P45452 1/20 0.41
CASP7 P55210 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17466005 0.83 MEN1 (0.58) GAAMEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL502194 0.82 SMN1; SMN2 (0.61) GAAMEN1KMT2ASMN1; SMN2SLC6A2
SCHEMBL6378903 0.80 MMP8 (0.50) GAASLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL27920341 0.80 SMN1; SMN2 (0.60) GAAMEN1KMT2ASMN1; SMN2SLC6A2
SCHEMBL11167719 0.80 PTGS1 (0.52) GAAMEN1KMT2ASMN1; SMN2CYP2D6
SCHEMBL5299951 0.79 SMN1; SMN2 (0.56) GAAMEN1KMT2ASMN1; SMN2MAPT
SCHEMBL17583661 0.79 CYP2D6 (0.52) GAASMN1; SMN2SLC6A2SLC6A4SLC6A3
SCHEMBL5878417 0.79 AKR1C3 (0.54) GAAKMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL15341770 0.79 AKR1C3 (0.54) GAAKMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL622042 0.79 L3MBTL1 (0.50) GAAMEN1KMT2ASMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313560-B1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION UNIV YALE (US) 2007-12-19 EP disclosed
EP-1313560-A4 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION UNIV YALE (US) 2005-02-09 EP disclosed
EP-1313560-A1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION YALE UNIVERSITY (US) 2003-05-28 EP disclosed
US-6562989-B2 Bicyclopentyl iron ligand and transition metal catalyst YALE UNIVERSITY 2003-05-13 US disclosed
US-20030008768-A1 Catalyst for aromatic C-O, C-N, and C-C bond formation NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-01-09 US disclosed
WO-2002011883-A1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION YALE UNIVERSITY (US) 2002-02-14 WO disclosed