SCHEMBL5282536

SCHEMBL5282536

Clc1cccc(-c2ccccc2)c1CBr

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.56
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.42
NPY1R P25929 1/20 0.42
NPY2R P49146 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
MAPK1 P28482 1/20 0.40
AKR1B1 P15121 1/20 0.39
MAOB P27338 2/20 0.38
CSNK2A1 P68400 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
MAPK14 Q16539 1/20 0.37
DPP4 P27487 3/20 0.37
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
HSD11B1 P28845 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5376614 0.85 ALDH1A1 (0.48) CYP2A6ALDH1A1MAPK1TAAR1DPP4
SCHEMBL9720402 0.82 CYP2A6 (0.58) CYP2A6ALDH1A1LMNANPY1RNPY2R
SCHEMBL10988341 0.80 CYP2A6 (0.56) CYP2A6ALDH1A1LMNANPY1RNPY2R
SCHEMBL27856687 0.80 CYP2A6 (0.56) CYP2A6ALDH1A1LMNANPY1RNPY2R
SCHEMBL28396527 0.78 CYP2A6 (0.54) CYP2A6ALDH1A1LMNANPY1RNPY2R
SCHEMBL11038800 0.78 CYP2A6 (0.43) CYP2A6ALDH1A1LMNANPY1RNPY2R
SCHEMBL31097818 0.78 CYP2A6 (0.54) CYP2A6ALDH1A1LMNANPY1RNPY2R
SCHEMBL5501718 0.78 ALDH1A1 (0.44) CYP2A6ALDH1A1MAPK1CSNK2A1DPP4
SCHEMBL9770 0.78 TAAR1 (0.50) CYP2A6ALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL5858344 0.78 DPP4 (0.47) CYP2A6ALDH1A1MAPK1DPP4PDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed
US-4536591-A Insecticidal [1,1'-biphenyl]-3-ylmethyl esters FMC CORPORATION (US) 1985-08-20 US disclosed
US-4507317-A Acaricidal 2,2'-bridged[1,1'-biphenyl]-3-ylmethyl esters FMC CORPORATION (US) 1985-03-26 US disclosed
US-4451484-A ALSO MITICIDES FMC CORPORATION (US) 1984-05-29 US disclosed
US-4433182-A Insecticidal 2,2'-bridged[1,1'-biphenyl]-3-ylmethyl esters FMC CORPORATION (US) 1984-02-21 US disclosed
US-4402973-A Insecticidal (1,1'-biphenyl)-3-ylmethyl esters FMC CORPORATION (US) 1983-09-06 US disclosed
US-4329518-A INSECTICIDES, ACARICIDES, MITICIDES FMC CORPORATION (US) 1982-05-11 US disclosed
EP-0049977-A1 Insecticidal (1,1'-biphenyl)-3-ylmethyl esters, their production and use and compositions containing them FMC Corporation (US) 1982-04-21 EP disclosed