SCHEMBL5283734

SCHEMBL5283734

COc1cccc(-c2ccc([N+](=O)[O-])c3onnc23)c1F

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 3/20 0.41
TDP1 Q9NUW8 2/20 0.40
ALDH1A1 P00352 1/20 0.40
RXFP1 Q9HBX9 2/20 0.38
LMNA P02545 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
POLB P06746 3/20 0.36
MAPT P10636 2/20 0.36
PIN1 Q13526 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
CASP3 P42574 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
DHODH Q02127 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788719 0.80 MEN1 (0.50) S1PR1TDP1ALDH1A1POLBHPGD
SCHEMBL7066582 0.73 LMNA (0.49) TDP1ALDH1A1LMNAL3MBTL1MAPT
SCHEMBL3203718 0.72 TDP1 (0.41) TDP1ALDH1A1LMNAL3MBTL1POLB
SCHEMBL11693495 0.70 TDP1 (0.67) TDP1ALDH1A1L3MBTL1MAPTNPC1
SCHEMBL2313725 0.66 TDP1 (0.46) TDP1ALDH1A1LMNAL3MBTL1MAPT
SCHEMBL31658972 0.66 GSTP1 (0.46) TDP1ALDH1A1L3MBTL1POLBMAPT
SCHEMBL2333611 0.66 TDP1 (0.41) TDP1ALDH1A1LMNAL3MBTL1POLB
SCHEMBL17209987 0.66 PARP1 (0.35) TDP1ALDH1A1LMNAPOLBMAPT
SCHEMBL626589 0.65 ALDH1A1 (0.53) TDP1ALDH1A1LMNAL3MBTL1POLB
SCHEMBL29524625 0.65 ALDH1A1 (0.53) TDP1ALDH1A1LMNAL3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758873-A1 UBIQUITIN LIGASE INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2007-03-07 EP disclosed
WO-2006002284-A1 UBIQUITIN LIGASE INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2006-01-05 WO disclosed