SCHEMBL5283777

SCHEMBL5283777

C[Si](C)(C)CCOCn1cc2c(N)cccc2n1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
TDP2 O95551 1/20 0.32
NSD2 O96028 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
BLM P54132 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PDE10A Q9Y233 2/20 0.31
DGAT1 O75907 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30546510 0.84 HDAC8 (0.36) NPC1PDE10ADGAT1
SCHEMBL30546525 0.81 NPC1 (0.35) NPC1
SCHEMBL4718492 0.79 ALDH1A1 (0.39) NPC1KDM4EMEN1ALDH1A1POLB
SCHEMBL29810321 0.79 NPC1 (0.35) NPC1
SCHEMBL27191935 0.78 PARP1 (0.35) NPC1PDE10ADGAT1
SCHEMBL10452108 0.77 NPC1 (0.36) NPC1ALDH1A1PDE10ADGAT1
SCHEMBL25239263 0.75 DGAT1 (0.33) NPC1MAPTDGAT1
SCHEMBL25323155 0.75 DGAT1 (0.37) NPC1PDE10ADGAT1
SCHEMBL6118775 0.75 ALDH1A1 (0.41) NPC1KDM4EMEN1TDP2NSD2
SCHEMBL3348756 0.74 MPO (0.46) NPC1KDM4EMEN1TDP2NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007085540-A1 1H-INDAZ0L-4-YL-2 , 4-PYRIMIDINEDIAMINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2007-08-02 WO disclosed
WO-2007028445-A1 6-INDOLYL-4-YL-AMINO-5-HALOGENO-2-PYRIMIDINYL-AMINO DERIVATIVES GLAXO GROUP LIMITED (GB) 2007-03-15 WO disclosed
WO-2007009681-A1 1 , 1-DIOXID0-2 , 3-DIHYDRO-l , 2-BENZISOTHIAZ0L-6-YL-1H-INDAZOL-4-YL-2 , 4-PYRIMIDINEDI AMINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2007-01-25 WO disclosed