SCHEMBL5284246

SCHEMBL5284246

O=C1c2ccc(OS(=O)(=O)C(F)(F)F)cc2CN1Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.46
GRM5 P41594 1/20 0.43
ACHE P22303 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ADAM17 P78536 1/20 0.41
HDAC4 P56524 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC6 Q9UBN7 1/20 0.41
NR3C1 P04150 1/20 0.40
CHRM5 P08912 1/20 0.40
CNR2 P34972 1/20 0.39
PARP1 P09874 1/20 0.39
PRMT5 O14744 2/20 0.39
WDR77 Q9BQA1 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4508979 0.88 GRM5 (0.58) GRM5ACHEPRMT5WDR77ITGB3
SCHEMBL1002943 0.82 ADAM17 (0.57) GRM5ACHEMEN1KMT2AADAM17
SCHEMBL2023150 0.76 GRM5 (0.50) GRM5ACHEMEN1KMT2AADAM17
SCHEMBL12581806 0.75 MEN1 (0.50) GRM5ACHEMEN1KMT2AHDAC4
SCHEMBL31409566 0.75 HDAC1 (0.49) GRM5ACHEMEN1KMT2AADAM17
SCHEMBL5282876 0.75 HDAC1 (0.49) GRM5ACHEMEN1KMT2AADAM17
SCHEMBL1500111 0.75 HDAC1 (0.49) GRM5ACHEMEN1KMT2AHDAC4
SCHEMBL3225584 0.75 GRM5 (0.49) GRM5ACHEMEN1KMT2AHDAC4
SCHEMBL19967154 0.74 DHPS (0.52) GRM5MEN1KMT2AHDAC4HDAC1
SCHEMBL12581703 0.74 GRM5 (0.46) GRM5ACHEMEN1KMT2AHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007000337-A1 BICYCLIC DERIVATIVES AS P38 KINASE INHIBITORS PALAU PHARMA, S.A. (ES) 2007-01-04 WO disclosed